| Manipulation of carrier proteins in antibiotic biosynthesis JJ La Clair, TL Foley, TR Schegg, CM Regan, MD Burkart Chemistry & biology 11 (2), 195-201, 2004 | 198 | 2004 |
| Site-specific protein modification: advances and applications TL Foley, MD Burkart Current opinion in chemical biology 11 (1), 12-19, 2007 | 137 | 2007 |
| Early drug discovery and development guidelines: for academic researchers, collaborators, and start-up companies J Strovel, S Sittampalam, NP Coussens, M Hughes, J Inglese, A Kurtz, ... Assay guidance manual [Internet], 2016 | 101 | 2016 |
| Targeting iron assimilation to develop new antibacterials TL Foley, A Simeonov Expert opinion on drug discovery 7 (9), 831-847, 2012 | 98 | 2012 |
| Discovery of trifluoromethyl glycol carbamates as potent and selective covalent monoacylglycerol lipase (MAGL) inhibitors for treatment of neuroinflammation LA McAllister, CR Butler, S Mente, SV O’Neil, KR Fonseca, JR Piro, ... Journal of medicinal chemistry 61 (7), 3008-3026, 2018 | 73 | 2018 |
| Azetidine and piperidine carbamates as efficient, covalent inhibitors of monoacylglycerol lipase CR Butler, EM Beck, A Harris, Z Huang, LA McAllister, CW Am Ende, ... Journal of Medicinal Chemistry 60 (23), 9860-9873, 2017 | 65 | 2017 |
| Assay guidance manual [Internet] S Markossian, A Grossman, K Brimacombe, M Arkin, D Auld, C Austin, ... Eli Lilly & Company and the National Center for Advancing Translational Sciences, 2004 | 64 | 2004 |
| An orthogonal active site identification system (OASIS) for proteomic profiling of natural product biosynthesis JL Meier, S Niessen, HS Hoover, TL Foley, BF Cravatt, MD Burkart ACS chemical biology 4 (11), 948-957, 2009 | 62 | 2009 |
| Discovery of ML324, a JMJD2 demethylase inhibitor with demonstrated antiviral activity G Rai, A Kawamura, A Tumber, Y Liang, JL Vogel, JH Arbuckle, NR Rose, ... Probe Reports from the NIH Molecular Libraries Program [Internet], 2013 | 53 | 2013 |
| Assay Guidance Manual: Quantitative Biology and Pharmacology in Preclinical Drug Discovery NP Coussens, GS Sittampalam, R Guha, K Brimacombe, A Grossman, ... Clinical and translational science 11 (5), 461-470, 2018 | 44 | 2018 |
| 4-(3-Chloro-5-(trifluoromethyl)pyridin-2-yl)-N-(4-methoxypyridin-2-yl)piperazine-1-carbothioamide (ML267), a Potent Inhibitor of Bacterial Phosphopantetheinyl … TL Foley, G Rai, A Yasgar, T Daniel, HL Baker, M Attene-Ramos, ... Journal of medicinal chemistry 57 (3), 1063-1078, 2014 | 44 | 2014 |
| A solution phase platform to characterize chemical reaction compatibility with DNA-encoded chemical library synthesis AS Ratnayake, ME Flanagan, TL Foley, JD Smith, JG Johnson, ... ACS combinatorial science 21 (10), 650-655, 2019 | 42 | 2019 |
| Probe reports from the NIH molecular libraries program G Rai, A Kawamura, A Tumber, Y Liang, JL Vogel, JH Arbuckle, NR Rose, ... National Center for Biotechnology Information, 2010 | 41 | 2010 |
| A strategy to discover inhibitors of Bacillus subtilis surfactin-type phosphopantetheinyl transferase A Yasgar, TL Foley, A Jadhav, J Inglese, MD Burkart, A Simeonov Molecular biosystems 6 (2), 365-375, 2010 | 41 | 2010 |
| Covalent Small Molecule Inhibitors of Ca2+-Bound S100B MC Cavalier, AD Pierce, PT Wilder, MJ Alasady, KG Hartman, DB Neau, ... Biochemistry 53 (42), 6628-6640, 2014 | 40 | 2014 |
| Phosphopantetheinyl transferase inhibition and secondary metabolism TL Foley, BS Young, MD Burkart The FEBS Journal 276 (23), 7134-7145, 2009 | 38 | 2009 |
| An optimized immunoaffinity fluorescent method for natural product target elucidation W Yu, G Guizzunti, TL Foley, MD Burkart, JJ La Clair Journal of natural products 73 (10), 1659-1666, 2010 | 37 | 2010 |
| Laetirobin from the Parasitic Growth of Laetiporus sulphureus on Robinia pseudoacacia MJ Lear, O Simon, TL Foley, MD Burkart, TJ Baiga, JP Noel, ... Journal of natural products 72 (11), 1980-1987, 2009 | 34 | 2009 |
| Selecting approaches for hit identification and increasing options by building the efficient discovery of actionable chemical matter from DNA-encoded libraries TL Foley, W Burchett, Q Chen, ME Flanagan, B Kapinos, X Li, ... SLAS DISCOVERY: Advancing the Science of Drug Discovery 26 (2), 263-280, 2021 | 28 | 2021 |
| Preparation of FRET reporters to support chemical probe development TL Foley, A Yasgar, CJ Garcia, A Jadhav, A Simeonov, MD Burkart Organic & biomolecular chemistry 8 (20), 4601-4606, 2010 | 28 | 2010 |
